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Дата публикации | Название | Авторы |
2021 | Dataset of NMR-Spectra Pyrrolyl- and Indolylazines and Evidence of Their Ability to Induce Heat Shock Genes Expression in Human Neurons | Dutysheva, E. A.; Utepova, I. A.; Trestsova, M. A.; Anisimov, A. S.; Charushin, V. N.; Chupakhin, O. N.; Margulis, B. A.; Guzhova, I. V.; Lazarev, V. F. |
2023 | Derivatives of 9-phosphorylated acridine as butyrylcholinesterase inhibitors with antioxidant activity and the ability to inhibit β-amyloid self-aggregation: potential therapeutic agents for Alzheimer’s disease | Makhaeva, G. F.; Kovaleva, N. V.; Rudakova, E. V.; Boltneva, N. P.; Lushchekina, S. V.; Astakhova, T. Y.; Timokhina, E. N.; Serebryakova, O. G.; Shchepochkin, A. V.; Averkov, M. A.; Utepova, I. A.; Demina, N. S.; Radchenko, E. V.; Palyulin, V. A.; Fisenko, V. P.; Bachurin, S. O.; Chupakhin, O. N.; Charushin, V. N.; Richardson, R. J. |
2021 | Design and Antioxidant Properties of Bifunctional 2H-Imidazole-Derived Phenolic Compounds-A New Family of Effective Inhibitors for Oxidative Stress-Associated Destructive Processes | Gerasimova, E. L.; Gazizullina, E. R.; Borisova, M. V.; Igdisanova, D. I.; Nikiforov, E. A.; Moseev, T. D.; Varaksin, M. V.; Chupakhin, O. N.; Charushin, V. N.; Ivanova, A. V. |
2022 | Development of Drugs with Direct Antiviral Action Based on Azaheterocyclic Systems | Charushin, V. N.; Rusinov, V. L.; Varaksin, M. V.; Chupakhin, O. N.; Kovtun, O. P.; Spasov, A. A. |
2017 | Diazatriphenylenes and their thiophene analogues: Synthesis and applications | Verbitskiy, E. V.; Rusinov, G. L.; Charushin, V. N. |
2020 | Dibenzo[ f,h]furazano[3,4- b]quinoxalines: Synthesis by Intramolecular Cyclization through Direct Transition Metal-Free C-H Functionalization and Electrochemical, Photophysical, and Charge Mobility Characterization | Kvashnin, Y. A.; Verbitskiy, E. V.; Eltsov, O. S.; Slepukhin, P. A.; Tameev, A. R.; Nekrasova, N. V.; Rusinov, G. L.; Nunzi, J. -M.; Chupakhin, O. N.; Charushin, V. N. |
2016 | Dihydroazolopyrimidine crownophanes. Synthesis and tuberculostatic activity | Ovchinnikova, I. G.; Valova, M. S.; Fedorova, O. V.; Tumashov, A. A.; Kravchenko, M. A.; Medvinsk′i, I. D.; Rusinov, G. L.; Charushin, V. N. |
2022 | DIRECT C-H/S-H COUPLING OF 2Н-IMIDAZOLE-1-OXIDES AND THIOPHENOLS IN THE SYNTHESIS OF PERSPEVTIVE AZAHETEROCYCLIC COMPOUNDS | Nikiforov, Е. A.; Vaskina, N. F.; Moseev, T. D.; Varaksin, M. V.; Charushin, V. N.; Chupakhin, O. N. |
2020 | Direct C-Li/C-H coupling of C6F5Li with azines and azoles N-oxides as efficient approach toward to polyfloorinated azaheterocycles | Moseev, T. D.; Varaksin, M. V.; Virlova, E. A.; Chupakhin, O. N.; Charushin, V. N. |
2022 | DIRECT C–H THIOLATION OF AZOLOPYRIMIDINES IN THE SYNTHESIS OF TRIAZAVIRIN® STRUCTURAL ANALOGUES | Silaeva, A. I.; Akulov, А. А.; Varaksin, М. V.; Charushin, V. N.; Rusinov, V. L. |
2019 | Direct Functionalization of C(sp 2 )-H Bond in Nonaromatic Azaheterocycles: Palladium-Catalyzed Cross-Dehydrogenative Coupling (CDC) of 2 H-Imidazole 1-Oxides with Pyrroles and Thiophenes | Akulov, A. A.; Varaksin, M. V.; Charushin, V. N.; Chupakhin, O. N. |
2016 | Direct Modification of Quercetin by 6-Nitroazolo[1,5-a]Pyrimidines | Gorbunov, E. B.; Rusinov, G. L.; Ulomskii, E. N.; El′tsov, O. S.; Rusinov, V. L.; Kartsev, V. G.; Charushin, V. N.; Khalymbadzha, I. A.; Chupakhin, O. N. |
2023 | (E)-2-(6-(4′-(Diphenylamino)-[1,1′-biphenyl]-2-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5(4H)-ylidene)-2-(6-(4′-(diphenylamino)-[1,1′-biphenyl]-2-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl)acetonitrile | Kvashnin, Y. A.; Slepukhin, P. A.; Gazizov, D. A.; Zhilina, E. F.; Rusinov, G. L.; Verbitskiy, E. V.; Charushin, V. N. |
2022 | Effect of the Silica–Magnetite Nanocomposite Coating Functionalization on the Doxorubicin Sorption/Desorption | Demin, A. M.; Vakhrushev, A. V.; Valova, M. S.; Korolyova, M. A.; Uimin, M. A.; Minin, A. S.; Pozdina, V. A.; Byzov, I. V.; Tumashov, A. A.; Chistyakov, K. A.; Levit, G. L.; Krasnov, V. P.; Charushin, V. N. |
2015 | Experimental comparative pharmacokinetics of levofloxacin, triazavirine, and related conjugate | Blazhennikova, I. V.; Kurpyakova, A. F.; Bykov, V. N.; Geibo, D. S.; Nikiforov, A. S.; Stepanov, A. V.; Charushin, V. N.; Chupakhin, O. N.; Kotovskaya, S. K.; Rusinov, V. L. |
2004 | Fluorinated Derivatives of Benz[4,5]imidazo[1,2-b][1,3] thiazole - Inhibitors of Reproduction of Measles Virus | Pokrovskii, A. G.; Il'Icheva, T. N.; Kotovskaya, S. K.; Romanova, S. A.; Charushin, V. N.; Chupakhin, O. N. |
2022 | Folic Acid Antimetabolites (Antifolates): A Brief Review on Synthetic Strategies and Application Opportunities | Kovalev, I. S.; Zyryanov, G. V.; Santra, S.; Majee, A.; Varaksin, M. V.; Charushin, V. N. |
2020 | Fragment-based approach to novel bioactive purine derivatives | Krasnov, V. P.; Levit, G. L.; Musiyak, V. V.; Gruzdev, D. A.; Charushin, V. N. |
2019 | Functionalized benzazines as luminescent materials and components for optoelectronics | Nosova, E. V.; Achelle, S.; Lipunova, G. N.; Charushin, V. N.; Chupakhin, O. N. |
2018 | An improved protocol for the preparation of 5, 11-dialkyl-6, 12-di(hetero)aryl-5, 11-dihydroindolo[3, 2-b]carbazoles and synthesis of their new 2, 8-dicyano-/2, 8-bis(benzo[d]thiazol-2-yl)-substituted derivatives | Irgashev, R. A.; Kazin, N. A.; Rusinov, G. L.; Charushin, V. N. |