Дата публикации | Название | Авторы |
2022 | 4-(Aryl)-Benzo[4,5]imidazo[1,2-a]pyrimidine-3-Carbonitrile-Based Fluorophores: Povarov Reaction-Based Synthesis, Photophysical Studies, and DFT Calculations | Fedotov, V. V.; Valieva, M. I.; Taniya, O. S.; Aminov, S. V.; Kharitonov, M. A.; Novikov, A. S.; Kopchuk, D. S.; Slepukhin, P. A.; Zyryanov, G. V.; Ulomsky, E. N.; Rusinov, V. L.; Charushin, V. N. |
2022 | 6-(Tetrazol-5-yl)-7-aminoazolo[1,5-a]pyrimidines as Novel Potent CK2 Inhibitors | Urakov, G. V.; Savateev, K. V.; Kotovskaya, S. K.; Rusinov, V. L.; Spasov, A. A.; Babkov, D. A.; Sokolova, E. V. |
2023 | Amino Derivatives of Diaryl Pyrimidines and Azolopyrimidines as Protective Agents against LPS-Induced Acute Lung Injury | Spasov, A.; Ovchinnikova, I.; Fedorova, O.; Titova, Y.; Babkov, D.; Kosolapov, V.; Borisov, A.; Sokolova, E.; Klochkov, V.; Skripka, M.; Velikorodnaya, Y.; Smirnov, A.; Rusinov, G.; Charushin, V. |
2022 | Azolo[1,5-a]pyrimidines and Their Condensed Analogs with Anticoagulant Activity | Savateev, K. V.; Fedotov, V. V.; Rusinov, V. L.; Kotovskaya, S. K.; Spasov, A. A.; Kucheryavenko, A. F.; Vasiliev, P. M.; Kosolapov, V. A.; Sirotenko, V. S.; Gaidukova, K. A.; Uskov, G. M. |
2022 | CK2 Inhibition and Antitumor Activity of 4,7-Dihydro-6-nitroazolo[1,5-a]pyrimidines | Lyapustin, D. N.; Kotovskaya, S. K.; Butorin, I. I.; Ulomsky, E. N.; Rusinov, V. L.; Babkov, D. A.; Pokhlebin, A. A.; Spasov, A. A.; Melekhin, V. V.; Tokhtueva, M. D.; Shcheglova, A. V.; Makeev, O. G. |
2022 | Discovery of Nitro-azolo[1,5-a]pyrimidines with Anti-Inflammatory and Protective Activity against LPS-Induced Acute Lung Injury | Spasov, A.; Kosolapov, V.; Babkov, D.; Klochkov, V.; Sokolova, E.; Miroshnikov, M.; Borisov, A.; Velikorodnaya, Y.; Smirnov, A.; Savateev, K.; Fedotov, V.; Kotovskaya, S.; Rusinov, V. |
2013 | Long-range 1H-15N J couplings providing a method for direct studies of the structure and azide-tetrazole equilibrium in a series of azido-1,2,4-triazines and azidopyrimidines | Shestakova, T. S.; Shenkarev, Z. O.; Deev, S. L.; Chupakhin, O. N.; Khalymbadzha, I. A.; Rusinov, V. L.; Arseniev, A. S. |
2013 | Microwave-assisted palladium-catalyzed C-C coupling versus nucleophilic aromatic substitution of hydrogen (SN H) in 5-bromopyrimidine by action of bithiophene and its analogues | Verbitskiy, E. V.; Cheprakova, E. M.; Zhilina, E. F.; Kodess, M. I.; Ezhikova, M. A.; Pervova, M. G.; Slepukhin, P. A.; Subbotina, J. O.; Schepochkin, A. V.; Rusinov, G. L.; Chupakhin, O. N.; Charushin, V. N. |
2023 | Novel Substituted Azoloazines with Anticoagulant Activity | Spasov, A. A.; Fedorova, O. V.; Rasputin, N. A.; Ovchinnikova, I. G.; Ishmetova, R. I.; Ignatenko, N. K.; Gorbunov, E. B.; Sadykhov, G. A. O.; Kucheryavenko, A. F.; Gaidukova, K. A.; Sirotenko, V. S.; Rusinov, G. L.; Verbitskiy, E. V.; Charushin, V. N. |
2022 | Searching for novel antagonists of adenosine A1 receptors among azolo[1,5-a]pyrimidine nitro derivatives | Yakovlev, D. S.; Vassiliev, P. M.; Agatsarskaya, Y. V.; Brigadirova, A. A.; Sultanova, K. T.; Skripka, M. O.; Spasov, A. A.; Savateev, K. V.; Rusinov, V. L.; Maltsev, D. V. |
2022 | Synthesis and Biological Investigation of 1,2,4-Triazolo[4,3- a ]azines as Potential HSF1 Inductors | Serebrennikova, P. O.; Utepova, I. A.; Chupakhin, O. N.; Guzhova, I. V.; Mikhaylova, E. R.; Antonchick, A. P. |
2022 | Synthesis of Pyrimidine Conjugates with 4-(6-Amino-hexanoyl)-7,8-difluoro-3,4-dihydro-3-methyl-2H-[1,4] benzoxazine and Evaluation of Their Antiviral Activity | Krasnov, V. P.; Musiyak, V. V.; Levit, G. L.; Gruzdev, D. A.; Andronova, V. L.; Galegov, G. A.; Orshanskaya, I. R.; Sinegubova, E. O.; Zarubaev, V. V.; Charushin, V. N. |